BDBM223320 KDOAM-25

SMILES CCN(CCN(C)C)C(=O)CNCc1cc(ccn1)C(N)=O

InChI Key InChIKey=PNFMVADNCOGWME-UHFFFAOYSA-N

Data  37 IC50  1 Kd

PDB links: 2 PDB IDs match this monomer.

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 223320   

TargetLysine-specific demethylase 6B(Homo sapiens (Human))
University of Oxford

LigandBDBM223320(KDOAM-25)Copy SMILESCopy InChI

Affinity DataIC50:  1.00E+5nMAssay Description:We previously described 4-carboxy-2-triazolopyridines as selective KDM2 inhibitors (England et al., 2014). In efforts to find alternative scaffolds b...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPurchasePC cidPC sidPDB

In DepthDetails ArticlePubMed
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